GROUP PUBLICATIONS

2024

79. Ziren Kong#, Zhu Li#, Junyi Chen#, Yixin Shi, Nan Li, Wenbin Ma, Yu Wang*, Zhi Yang*; Zhibo Liu*, A histogram of [18F]BBPA PET imaging differentiates non-neoplastic lesions from malignant brain tumors. EJNMMI Res. 2024, 14 (1).

78. Zhu Li#, Junyi Chen#, Ziren Kong, Yixin Shi, Mengxin Xu, Bo-Shuai Mu, Nan Li, Wenbin Ma, Zhi Yang, Yu Wang*; Zhibo Liu*, A bis-boron boramino acid PET tracer for brain tumor diagnosis. Eur J Nucl Med Mol Imag. 2024, 10.1007/s00259-024-06600-5.

77.  Jialing Sun#, Junyi Chen#, Yiming Sun, Yingqin Hou, Zhibo Liu*; Hua Lu*, On the origin of the low immunogenicity and biosafety of a neutral α-helical polypeptide as an alternative to polyethylene glycol. Bioact Mater. 2024, 32: 333-343.

76. Mengqi Chen#, Chunhong Wang#, Xuanyu Wang, Zhiyu Tu, Zexuan Ding, Zhibo Liu*An “AND” Logic-Gated Prodrug Micelle Locally Stimulates Antitumor ImmunityAdv Mater. 2024 36(6): 2307818.

 

2023

75. Di Sang, Keteng Lin, Yini Yang, Guangdi Ran, Bohan Li, Chen Chen, Qi Li, Yan Ma, Lihui Lu, Xi-Yang Cui, Zhibo Liu, Sheng-Qing Lv, Minmin Luo, Qinghua Liu, Yulong Li, Eric Erquan Zhang. Prolonged sleep deprivation induces a cytokine-storm-like syndrome in mammals. Cell. 2023,  186(25): 5500-5516.

74. Qunfeng Fu#, Siyong Shen#, Pengwei Sun, Zhi Gu, Yifei Bai, Xianglin Wang, Zhibo Liu*. Bioorthogonal chemistry for prodrug activation in vivo. Chem Soc Rev. 2023, 52: 7737-7772.

73. Hanbo Song#, Mengxin Xu#*, Jie Cai, Junyi Chen, Yu Liu, Qi Su, Zhu Li*, Zhibo Liu*. 225Ac-Labeled Antibody for Fibroblast Activation Protein-Targeted Alpha Therapy. Chemical & Biomedical Imaging. 2023, 1 (7): 628-636.

72. Mengxin Xu#, Junyi Chen#, Pu Zhang, Jie Cai, Hanbo Song, Zhu Li*, Zhibo Liu*. An antibody-radionuclide conjugate targets fibroblast activation protein for cancer therapy. Eur J Nucl Med Mol Imaging. 2023, 50: 3214–3224.

71. Yu Liu, Haocheng Tang, Tianchi Song, Mengxin Xu, Junyi Chen, Xi-Yang Cui, Yuxiang Han, Zhu Li, Zhibo Liu*. Organotrifluoroborate Enhances Tumor Targeting of Fibroblast Activation Protein Inhibitors for Targeted Radionuclide Therapy. Eur J Nucl Med Mol Imaging. 2023, 50: 2636–2646.

70. Yaxin Shi#, Zhibin Guo#, Qiang Fu#, Xinyuan Shen, Zhongming Zhang, Wenjia Sun, Jinqiang Wang, Junliang Sun, Zizhu Zhang, Tong Liu, Zhen Gu*, Zhibo Liu*Localized Nuclear Reaction Breaks Boron Drug Capsules Loaded with Immune Adjuvants for Cancer Immunotherapy. Nat Commun. 2023, 14: 1884.

69. Dongban Duan#, Yi Han#, Zhiyu Tu#, Haoxuan Guo, Zizhu Zhang, Yaxin Shi, Jiyuan Li, Qi Sun, Junyi Chen, Zhu Li, Tong Liu, Daqing Cui, Zhibo Liu*. Gadolinium Neutron Capture Reaction-Induced Nucleodynamic Therapy Potentiates Antitumor ImmunityCCS Chemistry. 2023, 5(11): 2589-2602.

68. Qi Sun#, Jiyuan Li#, Zexuan Ding, Zhibo Liu*. Radiopharmaceuticals heat anti-tumor immunity. Theranostics. 2023, 13(2): 767-786.

2022

67. 李嘉颢, 梁炜秋, 穆博帅, 刘志博*. 二氟甲基自由基反应及其在18F标记中的应用. 高等学校化学学报. 2022, 43(12), 20220652.

66. Qiang Wei, Yuhxuan Lee, Weiqiu Liang, Xiaolei Chen, Bo-Shuai Mu, Xi-Yang Cui, Wangsuo Wu, Shuming Bai, Zhibo Liu*. Photocatalytic Direct Borylation of Carboxylic AcidsNat Commun. 2022, 13: 7112.

65. Jie Ding*, Mengxin Xu*, Junyi Chen*, Pu Zhang, Li Huo*, Ziren Kong*, Zhibo Liu*. 86Y-Labeled Albumin-Binding Fibroblast Activation Protein Inhibitor for Late-Time-Point Cancer Diagnosis. Mol Pharm. 2022, 19(9): 3429−3438.

64. Zhibin Guo#, Hanyu Hong#, Yuedan Zheng, Ziyang Wang, Zexuan Ding, Qunfeng Fu, Zhibo Liu*. Radiotherapy-Induced Cleavage of Quaternary Ammonium Groups Activates Prodrugs in Tumors. Angew Chem Int Ed. 2022, 61(34): e202205014. 

63. Mengqi Chen, Chunhong Wang, Zexuan Ding, Hao Wang, Yu Wang, Zhibo Liu*A Molecular Logic Gate for Developing “AND” Logic Probes and the Application in Hepatopathy DifferentiationACS Central Science. 2022, 8: 837−844.

62. 陈俊艺, 刘宇, 徐梦欣, 刘志博*225Ac-213Bi发生器的制备与使用中华核医学与分子影像杂志2022, 42(6): 330-334. 

61. Xi-Yang Cui, Yu Liu, Changlun Wang, Zihao Wen, Yichen Li, Haocheng Tang, Juan Diwu, Yuchuan Yang, Mengchao Cui, Zhibo Liu*. China's Radiopharmaceuticals on Expressway: 2014-2021. Radiochimica Acta. 2022, https://doi.org/10.1515/ract-2021-1137.

60. Zexuan Ding, Zhibin Guo, Yuedan Zheng, Ziyang Wang, Qunfeng Fu, and Zhibo Liu*Radiotherapy reduces N-oxides for prodrug activation in tumors. J Am Chem Soc. 2022, 144(21):9458-9464.

59. Ziren Kong #, Zhu Li #, Junyi Chen #, Wenbin Ma, Yu Wang*, Zhi Yang*, Zhibo Liu*Larger 18F-fluoroboronotyrosine (FBY) active volume beyond MRI contrast enhancement in diffuse gliomas than in circumscribed brain tumors. EJNMMI Res. 2022, 12(1):22. 

58. Jiyuan Li#, Qi Sun#, Chuanjie Lu, Han Xiao, Zhibin Guo, Dongban Duan, Zizhu Zhang, Tong Liu, Zhibo Liu*Boron encapsulated in a liposome can be used for combinational neutron capture therapyNat Commun. 2022, 13: 2143.

57. Junyi Chen, Jingfeng Wang, MengXin Xu, Xianlu Jia, Guofang Song, Zhibo Liu*Production of positron-emitting radionuclide yttrium-86 with a computer-aided design target for positron emission tomographyNucl Med Biol. 2022, 108-109:54-60.

56. Junyi Chen, Mengxin Xu, Yu Liu, Dongban Duan, Yuxiang Han, Zhibo Liu*. Isolation of 212Pb from natural thorium for targeted alpha-therapyChin Chem Lett. 2022, 33(7):3474-3477.

55. Ziren Kong#, Zhu Li#, Junyi Chen#, Sirui Liu, Delin Liu, Jiyuan Li, Nan Li, Wenbin Ma, Feng Feng, Yu Wang*, Zhi Yang*, Zhibo Liu*. Metabolic characteristics of [18F] fluoroboronotyrosine (FBY) PET in malignant brain tumors. Nucl Med Biol. 2022, 106-107:80-87.

54. Mengxin Xu, Pu Zhang, Jie Ding, Junyi Chen, Li Huo, Zhibo Liu*. Albumin Binder–Conjugated Fibroblast Activation Protein Inhibitor Radiopharmaceuticals for Cancer TherapyJ Nucl Med. 2022, 63(6):952-958.

2021

53. 穆博帅, 徐洋, 刘志博*. 靶向PSMA放射性小分子药物研究进展同位素. 2021, 34 (6), 565-580.

52. Pu Zhang#, Mengxin Xu#, Jie Ding, Junyi Chen, Taiping Zhang, Li Huo*, Zhibo Liu*. Fatty acid-conjugated radiopharmaceuticals for fibroblast activation protein-targeted radiotherapyEur J Nucl Med Mol Imaging. 2021, 49, 1985–1996.

51. Huifang He, Jiyuan Li, Ping Jiang, Suqing Tian, Hao Wang, Ruitai Fan, Junqi Liu, Yuyan Yang, Zhibo Liu*. The basis and advances in clinical application of boron neutron capture therapyRadiat Oncol. 2021, 16(1):216.

50. Junyi Chen, Yinlong Lv, Feng Wang, Tianjue Zhang, Zhibo Liu*. Production and isolation of actinium-225 with a 100 MeV proton cyclotron and solid-phase extraction for targeted radiotherapy. Chemistry (HXTB). 2021, 84(11):1211-1219.

49. Chunhong Wang, Hanyu Hong, Mengqi Chen, Zexuan Ding, Yuchen Rui, Zi-Chen Li,Zhibo Liu*. Cationic Micelle as  In Vivo Catalyst for Tumor-Localized Cleavage Chemistry. Angew Chem Int Ed. 2021, 60, 19750-19758

48.Zhu Li#, Ziren Kong#, Junyi Chen, Jiyuan Li, Nan Li,  Zhi Yang*,Yu Wang*, Zhibo Liu*. 18F-Boramino Acid PET/CT in Healthy Volunteers and Glioma PatientsEur J Nucl Med Mol Imaging. 2021, 48(10):3113-3121.

47.Dongban Duan, Hao Dong, Zhiyu Tu, Chunhong Wang, Qunfeng Fu, Junyi Chen, Hai-peng Zhong, Ping Du, Ling-Dong Sun, Zhibo Liu*.  Desilylation Induced by Metal Fluoride Nanocrystals Enables Cleavage Chemistry In VivoJ Am Chem Soc2021, 143(5):2250-2255.

46.Jingyun Ren, Mengxin Xu, Junyi Chen, Jie Ding, Peipei Wang, Li Huo*, Fang Li*, Zhibo Liu*PET Imaging Facilitates Antibody Screening for Synergistic Radioimmunotherapy with A 177Lu-Labeled αPD-L1 Antibody. Theranostics. 2021, 11(1):304-315.

45.Liping Li, Kun Dai, Jiyuan Li, Yaxin Shi, Zizhu Zhang, Tong Liu, Ruiping Zhang*, Zhibo Liu*.  A Boron-10 Nitride Nanosheet for Combinational Boron Neutron Capture Therapy and Chemotherapy of Tumor.  Biomaterials2021, 268:120587.

2020

44.Yaxin Shi, Qiang Fu, Jiyuan Li, Zizhu Zhang, Hui Liu, Tong Liu, Zhibo Liu*.  A Covalent Organic Polymer as a Carborane Carrier for Imaging-Facilitated Boron Neutron Capture TherapyACS Appl Mater Interfaces. 2020, 12(50): 55564−55573.

43. 徐梦欣,  李一佳,  刘志博*细胞标记与体内追踪成像:在动物和人类中应用的最新进展. 中国组织工程研究2020, 24(19): 3108-3116.

42. Jiyuan Li, Zhiyu Tu, Zhibo Liu*走进曙色的冷门方向 :硼携带剂发展历程简述Scientia Sinica Chimica. 2020, 50: 1296–1319.

41.Qunfeng Fu, Hongyu Li, Dongban Duan, Changlun Wang, Huimin Ma, Zhibo Liu*External Radiation–Induced Local Hydroxylation Enables Remote Release of Functional Molecules in Tumors. Angew Chem Int Ed. 2020, 59(48): 21546–21552.

40.Qinyang Wang, Yupeng Wang, Jingjin Ding, Chunhong Wang, Xuehan Zhou, Wenqing Gao, Huanwei Huang, Feng Shao*, Zhibo Liu*. A Bioorthogonal System Reveals Antitumour Immune Function of Pyroptosis. Nature. 2020, 579, 421–426.

2019

39.Junyi Chen, Cong Li, Hanyu Hong, Hui Liu, Chunhong Wang, Mengxin Xu, Yuxiang Han, Zhibo Liu*Side Chain Optimization Remarkably Enhances the In Vivo Stability of 18F-Labeled Glutamine for Tumor Imaging. Mol Pharm. 2019,16, 12, 5035–5041.  

38.Qunfeng Fu, Junyi Chen,Zhibo Liu*Cherenkov Light: A New Light Source for Theranostics With Nano-Drug. J Nucl Radiochem. 2019: 41(2): 201-207.

37.Jiyuan Li, Yaxin Shi, Zizhu Zhang, Hui Liu, Lixin Lang, Tong Liu, Xiaoyuan Chen*, Zhibo Liu*. A Metabolically Stable Boron-Derived Tyrosine Serves as a Theranostic Agent for Positron Emission Tomography Guided Boron Neutron Capture TherapyBioconjug Chem. 2019, 30 (11), 2870-2878.

36.Liping Li, Jiyuan Li, Yaxin Shi, Ping Du, Zizhu Zhang, Tong Liu, Ruiping Zhang*, Zhibo Liu*. On-Demand Biodegradable Boron Nitride Nanoparticles for Positron Emission Tomography Guided Boron Neutron Capture Therapy. ACS Nano2019, 13 (12), 13843-13852.  

35.Hsiou-Ting Kuo, Mathieu Lepage, Kuo-Shyan Lin, Jinhe Pan, Zhengxing Zhang, Zhibo Liu, Alla Pryyma, Chengcheng Zhang, Helen Merkens, Aron Roxin, David Perrin, Francois Benard. One-step 18F-labeling and preclinical evaluation of prostate specific membrane antigen trifluoroborate probes for cancer imaging. J Nucl Med. 2019, 60(8), 1160-1166.
.

2018

34.Shi, Yaxin; Li, Jiyuan; Zhang, Zizhu; Duan, Dongban; Zhang, Zhengchu; Liu, Hui; Liu, Tong; Liu, Zhibo*Tracing Boron with Fluorescence and PET Imaging of Boronated Porphyrin Nanocomplex for Imaging Guided Boron Neutron Capture TherapyACS Appl Mater Interfaces. 2018, 10, 50, 43387-43395

33.Dongban Duan, Hui Liu, Mengxin Xu, Mengqi Chen, Yuxiang Han, Yaxin Shi, Zhibo Liu*Size-Controlled Synthesis of Drug Loaded Zeolitic Imidazolate Framework in Aqueous Solution and Size Impact on Their Cancer Theranostics In Vivo. ACS Appl Mater Interfaces​. 2018, 10(49): 42165-42174.

32.Cong Li, Hui Liu, Dongban Duan, Zhenhan Zhou, Zhibo Liu*Preclinical Study of An 18F-Labeled Glutamine Derivative for Cancer Imaging. Nucl Med Biol. 2018, 64: 34-40.

31.Mengxin Xu, Yuxiang Han, Guizhong Liu, Yang Xu, Dongban Duan, Hui Liu, Felix Du, Peter Luo, Zhibo Liu*Preclinical Study of A Fully Human Anti-PD-L1 Antibody as A Theranostic Agent for Cancer Immunotherapy. Mol Pharm. 2018, 15(10): 4426-4433.

30. Dongban Duan, Hui Liu, Yang Xu, Yuxiang Han, Mengxin Xu, Zhengchu Zhang, Zhibo Liu*Activating TiO2 Nanoparticles: Gallium-68 Serves as a High-Yield Photon Emitter for Cerenkov-Induced Photodynamic Therapy. ACS Appl Mater Interface. 2018, 10, 5278-5286.

29. Hui Liu, Yuxiang Han, Jiyuan Li, Ming Qin, Qunfeng Fu, Chunhong Wang, and Zhibo Liu*. (18)F-Alanine Derivative Serves as an ASCT2 Marker for Cancer Imaging. Mol Pharm. 2018, 15, 947-954.

28. Cong Li, Hui Liu, Yuxiang Han, Zhibo Liu*Nuclear Medicine: The Synergy of Radiochemistry and Molecular Medicine. University Chemistry. 2018, 33(3): 1-10.

27. Xiangyu Yang, Zhibo Liu, Huimin Zhang, Zhu Li, Jeeva P. Munasinghe, Gang Niu, Gaojun Teng, Xiaoyuan Chen. Preclinical evaluation of an (18)F-trifluoroborate methionine derivative for glioma imaging. Eur J Nucl Med Mol Imaging. 2018, 45, 585-592.

26.Feng Wang, Teli Liu, Liqiang Li, Xiaoyi Guo, Dongban Duan, Zhibo Liu, Hua Zhu, Zhi Yang. Production, quality control of next-generation PET radioisotope iodine-124 and its thyroid imaging. J Radioanal Nucl Chem2018, 318, 1999–2006.

2010-2017

25. Zhibo Liu*, Xiaoyuan Chen* Simple Bioconjugate Chemistry Serves Great Clinical Advances: Albumin as A Versatile Platform for Diagnosis and Precision Therapy. Chem Soc Rev, 2016, 45, 1432-1456 (*Coresponding author)

24. Zhibo Liu*, Haojun Chen, Kai Chen, Yihan Shao, Dale O. Kiesewetter, Gang Niu, Xiaoyuan Chen* Boramino Acid as A Marker for Amino Acid Transporter. Science Advances, 2015;1:e1500694 (*Coresponding authorhighlighted on C&EN News)

23. Zhibo Liu*, Kuo-Shyan Lin, François Bénard, Dale O. Kiesewetter, David M. Perrin*, Xiaoyuan Chen* A Broadly Applicable One-step 18F-Labeling Protocol with Organotrifluoroborates. Nat Protoc, 2015, 10, 1423–1432 (*Coresponding author)

22. Zhibo Liu, Guillaume Amouroux, Zhengxing Zhang, Nadine Colpo, Joseph Lau, David M. Perrin, Jinhe Pan, François Bénard, Navjit Hundal-Jabal, Kuo-Shyan Lin 18F-Trifluoroborate Derivatives of [Des-Arg10]Kallidin for Imaging Bradykinin B1 Receptor Expression with Positron Emission Tomography. Mol Pharm, 2015, 12, 974-982

21. Zhibo Liu, David M. Perrin, Using Principles of Physical Organic Chemistry to Designing Kinetically Stable Aryltrifluoroborates as 18F-Capture Agents for PET Imaging, J Phys Org Chem, 2015, 28, 210-214

20. Zhibo Liu, Daniel Chao, Ying Li, Richard Ting, Jihyoon Oh, David M. Perrin From Minutes to Years: Predicting Solvolysis Rates for Organotrifluoroborates, Chem Eur J, 2015, 21, 3924-3928

19. Zhibo Liu, Maral Pourghiasian, Gemma Dias, Joseph Lau, Francois Benard, Kuo-shyan Lin, David M. Perrin, An Organotrifluoroborate for Broadly Applicable One-Step 18F-Labeling, Angew Chem Int Ed, 2014, 53, 11876–11880 (Cover feature, highlighted on C&EN News)

18. Zhibo Liu, Mark Alex Radtke, May Q. Wong, Kuo-Shyan Lin, Donald Yapp, David M. Perrin, Dual Mode Fluorescent PET Tracers: Efficient modular synthesis of Rhodamine-[cRGD]2-Alkyl-18F-Trifluoroborate, Rapid 18F-labeling at very high specific activity, In vivo PET Imaging, and Ex vivo fluorescence, Bioconjugate Chem. 2014, 25, 1951–1962 (Cover feature)

17. Zhibo Liu, Maral Pourghiasian, Francois Benard, Jinhe Pan, Kuo-Shyan Lin, David M. Perrin, Preclinical Evaluation of A High Affinity 18F-Trifluorborate Octreotide Derivative for Somatostatin Receptor Imaging, J Nucl Med, 2014, 55, 1499-1505 (2014 JNM Editor's Choice Award)

16. Zhibo Liu, Navjit Hundal, May Q. Wong, Kuo-Shyan Lin, Donald Yapp, François Bénard, David M. Perrin, A New 18F-Heteroaryltrifluoroborate with Greatly Enhanced Stability That Is Labelled by 18F-19F-Isotope Exchange in Good Yield at High Specific Activity, Med Chem Comm, 2014, 5, 171–179

15. Zhibo Liu, Ying Li, Jerome Lozada, Paul Schaffer, Michael J. Adam, Thomas J. Ruth, David M. Perrin, Stoichiometric Leverage: Rapid 18F-Aryltrifluoroborate Radiosynthesis at Exceptionally High Specific Activity For Click Conjugation, Angew Chem Int Ed, 2013, 52, 2303-2307.

14. Zhibo Liu, Ying Li, Jerome Lozada, May Q. Wong, Jennifer Greene, Kuo-Shyan Lin, Donald Yapp, David M. Perrin, Kit-like 18F-labeling of RGD-19F-Arytrifluroborate in High Yield and at Extraordinarily High Specific Activity with Preliminary In Vivo Tumor Imaging, Nucl Med Biol, 2013, 40, 841-849.

13. Zhibo Liu, Ying Li, Jerome Lozada, Jinhe Pan, Kuo-Shyan Lin, Paul Schaffer, David M. Perrin, Rapid One-Step 18F-Labeling of Aryltrifluoroborate Conjugates by Isotope Exchange at High Specific Activity, J Labelled Comp Radiopharm., 2012, 55 491–496.

12. Joseph LauZhibo Liu, Kuo-Shyan Lin, Jinhe Pan, Zhengxing Zhang, Daniela Vullo, Claudiu T. Supuran, David M. Perrin, François Bénard Trimeric radiofluorinated sulfonamide derivatives to achieve in vivo selectivity for carbonic anhydrase IX-targeted PET imaging, J Nucl Med, 2015, 56, 1434-1440

11. Maral PourghiasianZhibo Liu, David M. Perrin, Jinhe Pan, Kuo-Shyan Lin, Francois Benard, 18F-AmBF3-MJ9: A novel radiofluorinated bombesin derivative for prostate cancer imaging, Bioorg Med Chem Lett, 2015, 23, 1500-1506

10. Jerome Lozada, Zhibo Liu, David M. Perrin, Base-promoted protodeboronation of 2,6-disubstituted arylboronic acids, J Org Chem, 2014, 79, 5365-5368

9. Ying Li, Zhibo Liu, Maral Pourghiasian, Kuo-Shyan Lin, Paul Schaffer, Francois Benard, David M. Perrin,Alkynyl-18F-ArBF3 for One-pot Click 18F-Labeling of Demobesin for In Vivo PET Imaging of Tumors Expressing the GRP-Receptor, Am J Nucl Med Mol Imaging, 2013, 3, 57-70.

8. Ying Li, Zhibo Liu, May Q. Wong, Kuo-Shyan Lin, Donald T. Yapp, David M. Perrin, One-Step 18F-Labeling of Dimeric CycloRGD at High Specific Activity for Functional PET Imaging of Tumors in Mice, Nucl Med Biol, 2013, 40, 959-966

7. Vadim Bernard-Gauthier, Justin J Bailey, Zhibo Liu, Björn Wängler, Carmen Wängler, Klaus Jurkschat, David M Perrin, Ralf Schirrmacher. From Unorthodox to Established: The Current Status of 18F-Trifluoroborate-and 18F-SiFA-Based Radiopharmaceuticals in PET Nuclear Imaging. Bioconjugate Chem., 2016, 27, 267–279

6. Zhengxing Zhang, Silvia Jenni, Chengcheng Zhang, Helen Merkens, Joseph Lau, Zhibo Liu, David M Perrin, François Bénard, Kuo-Shyan Lin Synthesis and evaluation of 18 F-trifluoroborate derivatives of triphenylphosphonium for myocardial perfusion imaging. Bioorg Med Chem Lett, 2016, 26, 1675–1679

5. Joseph Lau, Zhengxing Zhang, Silvia Jenni, Hsiou-Ting Kuo, Zhibo Liu, Daniela Vullo, Claudiu T Supuran, Kuo-Shyan Lin, Francois Benard PET Imaging of Carbonic Anhydrase IX Expression of HT-29 Tumor Xenograft Mice with 68Ga-Labeled Benzenesulfonamides Mol Pharm, 2016, 13, 1137–1146

4. Guillaume Amouroux, Jinhe Pan, Silvia Jenni, Chengcheng Zhang, Zhengxing Zhang, Navjit Hundal-Jabal, Nadine Colpo, Zhibo Liu, François Bénard, Kuo-Shyan Lin. Imaging Bradykinin B1 Receptor with 68Ga-Labeled [des-Arg10] Kallidin Derivatives: Effect of the Linker on Biodistribution and Tumor Uptake. Mol Pharmaceutics, 2015, 12, 2879–2888

3. Kuo-Shyan Lin, Guillaume Amouroux, Jinhe Pan, Zhengxing Zhang, Silvia Jenni, Joseph Lau, Zhibo Liu, François Bénard. Comparative Studies of Three 68Ga-Labeled [Des-Arg10] Kallidin Derivatives for Imaging Bradykinin B1 Receptor Expression with PET Imaging. J Nucl Med, 2015, 56(4), 622-627

2. Joseph Lau, Jinhe Pan, Zhengxing Zhang, Navjit Hundal-Jabal, Zhibo Liu, François Bénard, Kuo-Shyan Lin. Synthesis and evaluation of 18F-labeled tertiary benzenesulfonamides for imaging carbonic anhydrase IX expression in tumours with positron emission tomography. Bioorg Med Chem Lett, 2014, 24, 3064–3068

1. Jinhe Pan, Joseph Lau, Felix Mesak, Navjit Hundal, Maral Pourghiasian, Zhibo Liu, François Bénard, Shoukat Dedhar, Claudiu T. Supuran, and Kuo-Shyan Lin, Synthesis and evaluation of 18F-labeled carbonic anhydrase IX inhibitors for imaging with positron emission tomography, J Enzyme Inhib Med Chem, 2014, 29, 249-255